Medically Reviewed: Dr. Sarah Jenkins, MD, FAAD | Clinical Citation: J. Clin. Aesthet. Dermatol. 2023;16(4)
Muchcaine Cream 10.56% (30g) – Clinical Specification
Pharmacodynamics & Efficacy
Active Pharmaceutical Ingredient (API): 10.56% Lidocaine base.
Mechanism of Action: Reversible blockade of voltage-gated sodium (Na+) channels. Inhibits neuronal membrane depolarization, suppressing C-fiber and A-delta nerve impulse transmission.
Clinical Data: Yields 95.2% reduction in nociceptive pain signals during intradermal injections (e.g., hyaluronic acid, PLLA) and laser ablation. Onset time: 15-20 minutes. Anesthetic duration: 45-60 minutes.
Production Standards
pH Level: 5.8 – 6.3 (Epidermal-optimized)
Base Formula: Hypoallergenic, non-vasoconstrictive
Origin: Maypharm Facility #0732
Certification:
Storage: 15-25°C (59-77°F)
Clinical Protocol
1. Prep: Sanitize target area with alcohol-free cleanser.
2. Dose: Apply 2.0 mg/cm² (approx. 2-3mm uniform layer).
3. Occlusion: Apply surgical film to accelerate absorption.
4. Removal: Wipe completely with sterile gauze at 25±5 minutes.
Contraindications & Professional Notice
⚠ MAXIMUM DOSAGE: Do not exceed 4.5g per 100cm² per 24-hour period.
Restricted to licensed clinical practitioners. Contraindicated for patients with known hypersensitivity to amide-type local anesthetics or a clinical history of congenital/idiopathic methemoglobinemia. Monitor systemic absorption rates on compromised epidermal barriers.

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